Publication date: Available online 12 October 2023
Source: Bioorganic & Medicinal Chemistry
Author(s): Lennart Brewitz, H.T. Henry Chan, Petra Lukacik, Claire Strain-Damerell, Martin A. Walsh, Fernanda Duarte, Christopher J. Schofield
Monthly Archives: October 2023
Reading and erasing of histone crotonyllysine mimics by the AF9 YEATS domain and SIRT2 deacylase
Publication date: Available online 12 October 2023
Source: Bioorganic & Medicinal Chemistry
Author(s): Nurgül Bilgin, Vildan A. Türkmen, Nesrin Hammami, Nadja R. Christensen, Jordi C. J. Hintzen, Jasmin Mecinović
Editorial Board
Publication date: 30 October 2023
Source: Bioorganic & Medicinal Chemistry, Volume 94
Author(s):
Design, synthesis and antiplasmodial evaluation of new amide-, carbamate-, and ureido-type harmicines
Publication date: 30 October 2023
Source: Bioorganic & Medicinal Chemistry, Volume 94
Author(s): Marina Marinović, Hrvoje Rimac, Lais Pessanha de Carvalho, C. Rôla, S. Santana, Kristina Pavić, Jana Held, Miguel Prudêncio, Zrinka Rajić
Truxillic acid monoamides as fatty acid binding protein 5 inhibitors
Publication date: 30 October 2023
Source: Bioorganic & Medicinal Chemistry, Volume 94
Author(s): Chuanzhou Zhu, Livia Schutz, Kalani Jayanetti, Kathryn Takemura, Faniya Doswell, Liqun Wang, Iwao Ojima, Martin Kaczocha
Unraveling the unexpected aggregation behavior of Pyrazole-Based compounds Targeting Mycobacterium tuberculosis UDP-Galactopyranose mutase
Publication date: 30 October 2023
Source: Bioorganic & Medicinal Chemistry, Volume 94
Author(s): Dalia M. Ahmed, David A.R. Sanders
Design and synthesis of sulfonamides incorporating a biotin moiety: Carbonic anhydrase inhibitory effects, antiproliferative activity and molecular modeling studies
Publication date: 30 October 2023
Source: Bioorganic & Medicinal Chemistry, Volume 94
Author(s): Paloma Begines, Alessandro Bonardi, Alessio Nocentini, Paola Gratteri, Simone Giovannuzzi, Roberto Ronca, Camilla Tavani, Maria Luisa Massardi, Óscar López, Claudiu T. Supuran
Discovery of potential novel TRPC5 inhibitors by virtual screening and bioassay
Publication date: 30 October 2023
Source: Bioorganic & Medicinal Chemistry, Volume 94
Author(s): Meiling Shen, Lingfeng Li, Yue Li, Xi Gu, Longhui Bai, Chengfeng Xia, Wenyong Xiong, Zhili Zuo
Design of a structure-activity relationship model of vitamin K epoxide reductase (VKORC1) inhibitors combining chemical synthesis of new compounds, enzymatic assays and molecular modelling
Publication date: 30 October 2023
Source: Bioorganic & Medicinal Chemistry, Volume 94
Author(s): Nolan Chatron, Manon Boulven, Adrien Montagut-Romans, Flavien Ponsot, Maïwenn Jacolot, Hervé Caruel, Etienne Benoît, Florence Popowycz, Virginie Lattard
Pentacyclic triterpene-amino acid derivatives induced apoptosis and autophagy in tumor cells, affected the JNK and PI3K/AKT/mTOR pathway
Publication date: 30 October 2023
Source: Bioorganic & Medicinal Chemistry, Volume 94
Author(s): Li-qiong Zhang, Li Sun, Yu-qing Zhou, Jing-jing Liu, Quan-de Wang, Wei-bin Mo, Ke-guang Cheng