Publication date: 5 December 2023
Source: European Journal of Medicinal Chemistry, Volume 261
Author(s): Tingkai Chen, Xu Tang, Zhenqi Wang, Feng Feng, Chunlei Xu, Qun Zhao, Yulan Wu, Haopeng Sun, Yao Chen
Monthly Archives: October 2023
Targeted protein degradation in drug development: Recent advances and future challenges
Publication date: 5 December 2023
Source: European Journal of Medicinal Chemistry, Volume 261
Author(s): Jian Song, Mingzheng Hu, Jun Zhou, Songbo Xie, Tianliang Li, Yan Li
Antiparasitic activity of ivermectin: Four decades of research into a “wonder drug”
Publication date: 5 December 2023
Source: European Journal of Medicinal Chemistry, Volume 261
Author(s): Michał Sulik, Michał Antoszczak, Adam Huczyński, Dietmar Steverding
Synthesis and clinical application of small-molecule inhibitors of Janus kinase
Publication date: 5 December 2023
Source: European Journal of Medicinal Chemistry, Volume 261
Author(s): Jing-Yi Zhang, Jin-Feng Sun, Peng Nie, Piet Herdewijn, Ya-Tao Wang
Synthetic approaches and application of clinically approved small-molecule Anti-HIV drugs: An update
Publication date: 5 December 2023
Source: European Journal of Medicinal Chemistry, Volume 261
Author(s): Lu Sun, Peng Nie, Li Luan, Piet Herdewijn, Ya-Tao Wang
Recent advances of antitumor leading compound Erianin: Mechanisms of action and structural modification
Publication date: 5 December 2023
Source: European Journal of Medicinal Chemistry, Volume 261
Author(s): Lu Ma, Menglong Li, Yueteng Zhang, Kangdong Liu
Identification of 1,3,4-oxadiazolyl-containing β-carboline derivatives as novel α-glucosidase inhibitors with antidiabetic activity
Publication date: 5 December 2023
Source: European Journal of Medicinal Chemistry, Volume 261
Author(s): Di Xiao, Li Lu, Bingwen Liang, Zhuang Xiong, Xuetao Xu, Wen-Hua Chen
Synthesis of bitopic ligands based on fallypride and evaluation of their affinity and selectivity towards dopamine D<sub>2</sub> and D<sub>3</sub> receptors
Publication date: 5 December 2023
Source: European Journal of Medicinal Chemistry, Volume 261
Author(s): Gui-Long Tian, Chia-Ju Hsieh, Michelle Taylor, Ji Youn Lee, Aladdin A. Riad, Robert R. Luedtke, Robert H. Mach
Identification of novel dithiocarbamate-copper complexes targeting p97/NPL4 pathway in cancer cells
Publication date: 5 December 2023
Source: European Journal of Medicinal Chemistry, Volume 261
Author(s): Martin Loffelmann, Zdeněk Škrott, Dušana Majera, Pavel Štarha, Vladimír Kryštof, Martin Mistrík
Novel chlorin e<sub>6</sub>-based conjugates of tyrosine kinase inhibitors: Synthesis and photobiological evaluation as potent photosensitizers for photodynamic therapy
Publication date: 5 December 2023
Source: European Journal of Medicinal Chemistry, Volume 261
Author(s): Fei Huang, Yu Li, Xing-Jie Zhang, Mei-Yu Lin, Gui-Yan Han, Hui-Ying Lin, Hui-Yun Lin, Zhenyuan Miao, Bu-Hong Li, Chun-Quan Sheng, Jian-Zhong Yao