Copper-Catalyzed Intramolecular Dearomative Aza-Wacker Reaction of Indole

Chem. Commun., 2024, Accepted Manuscript
DOI: 10.1039/D3CC06217A, Communication
Bi Wang, Ren-Xiao Liang, Zhenlu Shen, Yi-Xia Jia
Herein, we describe a copper-catalyzed intramolecular dearomative amination of indoles via a formal aza-Wacker reaction. This protocol provides an efficient method to access aza-polycyclic indoline molecules bearing exocyclic C=C bonds...
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