Chem. Sci., 2023, 14,10800-10805
DOI: 10.1039/D3SC04083F, Edge Article
DOI: 10.1039/D3SC04083F, Edge Article


Jessica Iegre, Sona Krajcovicova, Anders Gunnarsson, Lisa Wissler, Helena Käck, Anna Luchniak, Stefan Tångefjord, Frank Narjes, David R. Spring
Application of DVP stapling methodology to efficiently develop Nrf2 peptides with nM activity in enzymatic assays, submicromolar activity in cells and non-cytotoxicity, characterised by high resolution X-ray co-crystallography.
The content of this RSS Feed (c) The Royal Society of Chemistry
Application of DVP stapling methodology to efficiently develop Nrf2 peptides with nM activity in enzymatic assays, submicromolar activity in cells and non-cytotoxicity, characterised by high resolution X-ray co-crystallography.
The content of this RSS Feed (c) The Royal Society of Chemistry