Publication date: Available online 20 February 2023
Source: Bioorganic & Medicinal Chemistry Letters
Author(s): Yaling He, Dong Liu, Changsong Zhu, Xue Chen, Hongling Ye, Ming Ye
Category Archives: Bioorganic & Medicinal Chemistry Letters
Amphiphilic tribasic galactosamines potentiate rifampicin in Gram-negative bacteria at low Mg<sup>++</sup>/Ca<sup>++</sup>concentrations
Publication date: Available online 8 June 2023
Source: Bioorganic & Medicinal Chemistry Letters
Author(s): Ayan Mukherjee, Danyel Ramirez, Rajat Arora, Gilbert Arthur, Frank Schweizer
Design and Synthesis of a Library of C2-Substituted Sulfamidoadenosines to Probe Bacterial Permeability
Publication date: Available online 20 September 2023
Source: Bioorganic & Medicinal Chemistry Letters
Author(s): Shibin Zhao, Julian Maceren, Mia Chung, Samantha Stone, Raphael Geißen, Melissa S. Boby, Bradley S. Sherborne, Derek S. Tan
Development of small molecule inhibitors of natural killer group 2D receptor (NKG2D)
Publication date: Available online 29 September 2023
Source: Bioorganic & Medicinal Chemistry Letters
Author(s): Jocelyn Wang, Kohki M. Nakafuku, Jeannie Ziff, Christine F. Gelin, Hadi Gholami, Aaron A. Thompson, Nathan K. Karpowich, Luis Limon, Heather R. Coate, Kelly L. Damm-Ganamet, Amy Y. Shih, Joanna C. Grant, Marjorie Côte, Puiying A. Mak, Heather A. Pascual, Marie-Laure Rives, James P. Edwards, Jennifer D. Venable, Hariharan Venkatesan, Zhicai Shi
Benzyl stapled modification and anticancer activity of antimicrobial peptide A4K14-Citropin 1.1
Publication date: Available online 6 October 2023
Source: Bioorganic & Medicinal Chemistry Letters
Author(s): Huaxing Shen, Nan Zhang, Xianglong Kong, Nan Wang, Hong-Gang Hu, Wei Cong, Chao Liu
5-HT<sub>6</sub> receptor antagonists. Design, synthesis, and structure–activity relationship of substituted 2-(1-methyl-4-piperazinyl)pyridines
Publication date: Available online 6 October 2023
Source: Bioorganic & Medicinal Chemistry Letters
Author(s): Michał Gałęzowski, Charles-Henry Fabritius, Ullamari Pesonen, Harri Salo, Marta Olszak-Płachta, Klaudia Czerwińska, Justyna Adamczyk, Marcin Król, Peteris Prusis, Magdalena Sieprawska-Lupa, Maciej Mikulski, Katja Kuokkanen, Radosław Obuchowicz, Timo Korjamo, Niina Jalava, Agnieszka Nikiforuk, Mateusz Nowak
Short synthesis of a broadly Reactive, cell permeable serine hydrolase Fluorophosphonate-Alkyne probe
Publication date: 15 October 2023
Source: Bioorganic & Medicinal Chemistry Letters, Volume 95
Author(s): Srihari Konduri, Joshua Schweer, Dionicio Siegel
Design, synthesis and biological evaluation of chalcone derivatives as potent and orally active hCYP3A4 inhibitors
Publication date: 15 October 2023
Source: Bioorganic & Medicinal Chemistry Letters, Volume 95
Author(s): Shiwei Lu, Feng Zhang, Jiahao Gong, Jian Huang, Guanghao Zhu, Yitian Zhao, Qi Jia, Yiming Li, Bo Li, Kaixian Chen, Weiliang Zhu, Guangbo Ge
Design, synthesis and antitumor effects of novel benzimidazole derivatives as PI3K inhibitors
Publication date: 15 October 2023
Source: Bioorganic & Medicinal Chemistry Letters, Volume 95
Author(s): Wenping Wu, Sisi Li, Junjie Chen, Tena Duo, Cheng Ma
Design, synthesis, and biological evaluation of THIQ as antidepressive agents
Publication date: 15 October 2023
Source: Bioorganic & Medicinal Chemistry Letters, Volume 95
Author(s): Xiaopeng Wei, Man Zhang, Yijing Guo, Qianqian Chang, Wei Qiao