Publication date: 5 December 2023
Source: European Journal of Medicinal Chemistry, Volume 261
Author(s): Shankar Gupta, Gurkaran Singh Baweja, Shamsher Singh, Mehdi Irani, Rajveer Singh, Vivek Asati
Category Archives: European Journal of Medicinal Chemistry
Synthesis of cell penetrating peptide sterol coupler and its liposome study on S-mRNA
Publication date: 5 December 2023
Source: European Journal of Medicinal Chemistry, Volume 261
Author(s): Yuan Li, Wenlin Ma, Wen Su, Zhihong Yan, Lin Jia, Jie Deng, Ali Zhu, Yanbo Xie, Xinyi Li, Wanhui Shao, Yuman Ma, Linze Che, Tao Zhu, Haomeng Wang, Mingyuan Li, Peng Yu
Synthesis and biological evaluation of fluoroquinolones containing a pyridoxine derivatives moiety
Publication date: 5 December 2023
Source: European Journal of Medicinal Chemistry, Volume 261
Author(s): Nikita V. Shtyrlin, Airat R. Kayumov, Maria N. Agafonova, Marsel R. Garipov, Alina E. Gatina, Mikhail V. Pugachev, Elena S. Bulatova, Denis Y. Grishaev, Alfiya G. Iksanova, Rail M. Khaziev, Ilnur M. Ganiev, Aleksandr M. Aimaletdinov, Oleg I. Gnezdilov, Yurii G. Shtyrlin
Synthesis of bitopic ligands based on fallypride and evaluation of their affinity and selectivity towards dopamine D<sub>2</sub> and D<sub>3</sub> receptors
Publication date: 5 December 2023
Source: European Journal of Medicinal Chemistry, Volume 261
Author(s): Gui-Long Tian, Chia-Ju Hsieh, Michelle Taylor, Ji Youn Lee, Aladdin A. Riad, Robert R. Luedtke, Robert H. Mach
Identification of novel dithiocarbamate-copper complexes targeting p97/NPL4 pathway in cancer cells
Publication date: 5 December 2023
Source: European Journal of Medicinal Chemistry, Volume 261
Author(s): Martin Loffelmann, Zdeněk Škrott, Dušana Majera, Pavel Štarha, Vladimír Kryštof, Martin Mistrík
Novel chlorin e<sub>6</sub>-based conjugates of tyrosine kinase inhibitors: Synthesis and photobiological evaluation as potent photosensitizers for photodynamic therapy
Publication date: 5 December 2023
Source: European Journal of Medicinal Chemistry, Volume 261
Author(s): Fei Huang, Yu Li, Xing-Jie Zhang, Mei-Yu Lin, Gui-Yan Han, Hui-Ying Lin, Hui-Yun Lin, Zhenyuan Miao, Bu-Hong Li, Chun-Quan Sheng, Jian-Zhong Yao
The design, synthesis, and inhibition of <em>Clostridioides difficile</em> spore germination by acyclic and bicyclic tertiary amide analogs of cholate
Publication date: 5 December 2023
Source: European Journal of Medicinal Chemistry, Volume 261
Author(s): Shiv K. Sharma, Angel R. Schilke, Jacqueline R. Phan, Christopher Yip, Prateek V. Sharma, Ernesto Abel-Santos, Steven M. Firestine
Synthesis and mechanism of action of new purine derivatives against triple negative breast cancer
Publication date: 5 December 2023
Source: European Journal of Medicinal Chemistry, Volume 261
Author(s): Qian Zhang, Guoyang Sun, Yuna Huang, Shanshan Cui, Tingshen Li, Lianbo Zhao, Kui Lu, Peng Yu, Yongmin Zhang, Herve Galons, Nassima Oumata, Yuou Teng
Fragment-based and structure-guided discovery of perforin inhibitors
Publication date: 5 December 2023
Source: European Journal of Medicinal Chemistry, Volume 261
Author(s): Jiney Jose, Ruby H.P. Law, Eleanor W.W. Leung, Dorothy C.C. Wai, Hedieh Akhlaghi, Indu R. Chandrashekaran, Tom T. Caradoc-Davies, Ilia Voskoboinik, John Feutrill, David Middlemiss, Devadharshini Jeevarajah, Tanya Bashtannyk-Puhalovich, Anna C. Giddens, Tet Woo Lee, Stephen M.F. Jamieson, Joseph A. Trapani, James C. Whisstock, Julie A. Spicer, Raymond S. Norton
A dipyridophenazine Ni(II) dithiolene complex as a dual-acting cancer phototherapy agent activatable within the phototherapeutic window
Publication date: 5 December 2023
Source: European Journal of Medicinal Chemistry, Volume 261
Author(s): Tukki Sarkar, Somarupa Sahoo, Suditi Neekhra, Milan Paul, Swati Biswas, Bathini Nagendra Babu, Rohit Srivastava, Akhtar Hussain