Discovery of novel multifunctional ligands targeting GABA transporters, butyrylcholinesterase, β-secretase, and amyloid β aggregation as potential treatment of Alzheimer’s disease

Publication date: 5 December 2023

Source: European Journal of Medicinal Chemistry, Volume 261

Author(s): Paula Zaręba, Kamil Łątka, Gabriela Mazur, Beata Gryzło, Anna Pasieka, Justyna Godyń, Dawid Panek, Anna Skrzypczak-Wiercioch, Georg C. Höfner, Gniewomir Latacz, Maciej Maj, Alba Espargaró, Raimon Sabaté, Krzysztof Jóźwiak, Klaus T. Wanner, Kinga Sałat, Barbara Malawska, Katarzyna Kulig, Marek Bajda

Design, synthesis, and biological evaluation of quinoline-piperazine/pyrrolidine derivatives as possible antileishmanial agents

Publication date: 5 December 2023

Source: European Journal of Medicinal Chemistry, Volume 261

Author(s): Sarita Katiyar, Karthik Ramalingam, Abhishek Kumar, Alisha Ansari, Amol Chhatrapati Bisen, Garvita Mishra, Sachin Nashik Sanap, Rabi Sankar Bhatta, Bidyut Purkait, Neena Goyal, Koneni V. Sashidhara