Development of small molecule inhibitors of natural killer group 2D receptor (NKG2D)

Publication date: Available online 29 September 2023

Source: Bioorganic & Medicinal Chemistry Letters

Author(s): Jocelyn Wang, Kohki M. Nakafuku, Jeannie Ziff, Christine F. Gelin, Hadi Gholami, Aaron A. Thompson, Nathan K. Karpowich, Luis Limon, Heather R. Coate, Kelly L. Damm-Ganamet, Amy Y. Shih, Joanna C. Grant, Marjorie Côte, Puiying A. Mak, Heather A. Pascual, Marie-Laure Rives, James P. Edwards, Jennifer D. Venable, Hariharan Venkatesan, Zhicai Shi

5-HT<sub>6</sub> receptor antagonists. Design, synthesis, and structure–activity relationship of substituted 2-(1-methyl-4-piperazinyl)pyridines

Publication date: Available online 6 October 2023

Source: Bioorganic & Medicinal Chemistry Letters

Author(s): Michał Gałęzowski, Charles-Henry Fabritius, Ullamari Pesonen, Harri Salo, Marta Olszak-Płachta, Klaudia Czerwińska, Justyna Adamczyk, Marcin Król, Peteris Prusis, Magdalena Sieprawska-Lupa, Maciej Mikulski, Katja Kuokkanen, Radosław Obuchowicz, Timo Korjamo, Niina Jalava, Agnieszka Nikiforuk, Mateusz Nowak